5.05772
Pirenzepine Dihydrochloride
Synonym(s):
Pirenzepine Dihydrochloride, Muscarinic Acetylcholine Receptor (mAChR) M1 Antagonist, Pirenzepine dihydrochloride
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About This Item
Empirical Formula (Hill Notation):
C19H21N5O2 · 2HCl
CAS Number:
Molecular Weight:
424.32
MDL number:
UNSPSC Code:
12352200
NACRES:
NA.77
Assay:
≥99% (HPLC)
Form:
solid
Storage condition:
OK to freeze, protect from light
assay
≥99% (HPLC)
Quality Segment
form
solid
manufacturer/tradename
Calbiochem®
storage condition
OK to freeze, protect from light
color
white
solubility
water: 100 mM
storage temp.
2-8°C
SMILES string
N4(CCN(CC4)C)CC(=O)[n]1c2ncccc2[nH][c](c3c1cccc3)=O
InChI
1S/C19H21N5O2/c1-22-9-11-23(12-10-22)13-17(25)24-16-7-3-2-5-14(16)19(26)21-15-6-4-8-20-18(15)24/h2-8H,9-13H2,1H3,(H,21,26)
InChI key
RMHMFHUVIITRHF-UHFFFAOYSA-N
General description
An antagonist selective for mAChR subtype M1. Used for studying the functional roles of M1 receptors in both central and peripheral nervous systems.
Biochem/physiol Actions
Primary Target
M1
M1
Preparation Note
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Other Notes
Shirey, K., et al., 2009. J. Neurosci.29, 14271.
Pelat, M., et al., 1999. Eur.J. Pharmacol.379, 117.
Burford NT, et al. 1996. Biochem. J.315, 883.
Pelat, M., et al., 1999. Eur.J. Pharmacol.379, 117.
Burford NT, et al. 1996. Biochem. J.315, 883.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Disclaimer
Toxicity: Standard Handling (A)
Storage Class
11 - Combustible Solids
wgk
WGK 2
flash_point_f
Not applicable
flash_point_c
Not applicable
Certificates of Analysis (COA)
Search for Certificates of Analysis (COA) by entering the products Lot/Batch Number. Lot and Batch Numbers can be found on a product’s label following the words ‘Lot’ or ‘Batch’.
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