Skip to Content
Merck
CN

539636

PKCθ Pseudosubstrate Inhibitor, Myristoylated

The PKCθ Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKCθ. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

Synonym(s):

PKCθ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH2, Protein Kinase C θ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH2, Protein Kinase Cθ Pseudosubstrate Inhibitor, Myristoylated

Sign In to View Organizational & Contract Pricing.

Select a Size

About This Item

Empirical Formula (Hill Notation):
C105H182N35O22S
Molecular Weight:
2318.85
NACRES:
NA.77
UNSPSC Code:
12352200

Key Documents

View All Documentation
Technical Service
Need help? Our team of experienced scientists is here for you.
Let Us Assist
Technical Service
Need help? Our team of experienced scientists is here for you.
Let Us Assist

Product Name

PKCθ Pseudosubstrate Inhibitor, Myristoylated, The PKCθ Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKCθ. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

assay

≥95% (HPLC)

form

lyophilized solid

manufacturer/tradename

Calbiochem®

storage condition

OK to freeze
desiccated (hygroscopic)

solubility

water: 2 mg/mL

shipped in

ambient

storage temp.

−20°C

Quality Level

100

Related Categories

Disclaimer

Toxicity: Standard Handling (A)

Biochem/physiol Actions

Reversible: yes
Primary Target
protein kinase Cθ
Product competes with ATP.
Cell permeable: yes

General description

A cell-permeable, reversible, substrate competitive, myristoylated form of the inhibitor of protein kinase Cθ isozyme pseudosubstrate inhibitor (Cat. No. 539634).
Cell-permeable myristoylated protein kinase Cq pseudosubstrate sequence peptide (Cat. No. 539634). Useful for studies of PKCθ function in intact cells. Sold on the basis of peptide content.

Other Notes

Myr-Leu-His-Gln-Arg-Arg-Gly-Ala-Ile-Lys-Gln-Ala-Lys-Val-His-His-Val-Lys-Cys-NH₂
Osada, S., et al. 1992. Mol. Cell Biol.12, 3930.

Physical form

Supplied as a trifluoroacetate salt.

Preparation Note

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for 6 months at -20°C.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Storage Class

11 - Combustible Solids

wgk

WGK 1

flash_point_f

Not applicable

flash_point_c

Not applicable

Certificates of Analysis (COA)

Search for Certificates of Analysis (COA) by entering the products Lot/Batch Number. Lot and Batch Numbers can be found on a product’s label following the words ‘Lot’ or ‘Batch’.

Already Own This Product?

Find documentation for the products that you have recently purchased in the Document Library.

Visit the Document Library

Our team of scientists has experience in all areas of research including Life Science, Material Science, Chemical Synthesis, Chromatography, Analytical and many others.

Contact Technical Service