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SML0299

Biphalin trifluoroacetate salt

≥97% (HPLC)

别名:

1,2-Bis(L-Tyr-D-Ala-Gly-L-Phe-)hydrazine, L-Tyrosyl-D-alanylglycyl-L-phenylalanine 2-(L-tyrosyl-D-alanylglycyl-L-phenylalanyl)hydrazide

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关于此项目

经验公式（希尔记法）:
C46H56N10O10 · xC2HF3O2
化学文摘社编号:
126872-95-5
分子量:
909.00 (free base basis)
NACRES:
NA.77
PubChem Substance ID:
329825305
UNSPSC Code:
12352200
MDL number:
MFCD23380198
Assay:
≥97% (HPLC)
Form:
lyophilized solid
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Quality Segment

100

assay

≥97% (HPLC)

form

lyophilized solid

color

white to beige

shipped in

wet ice

storage temp.

−20°C

SMILES string

OC(=O)C(F)(F)F.C[C@@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](Cc2ccccc2)C(=O)NNC(=O)[C@H](Cc3ccccc3)NC(=O)CNC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc4ccc(O)cc4

InChI

1S/C46H56N10O10.C2HF3O2/c1-27(51-43(63)35(47)21-31-13-17-33(57)18-14-31)41(61)49-25-39(59)53-37(23-29-9-5-3-6-10-29)45(65)55-56-46(66)38(24-30-11-7-4-8-12-30)54-40(60)26-50-42(62)28(2)52-44(64)36(48)22-32-15-19-34(58)20-16-32;3-2(4,5)1(6)7/h3-20,27-28,35-38,57-58H,21-26,47-48H2,1-2H3,(H,49,61)(H,50,62)(H,51,63)(H,52,64)(H,53,59)(H,54,60)(H,55,65)(H,56,66);(H,6,7)/t27-,28-,35+,36+,37+,38+;/m1./s1

InChI key

KNKVMVJCRGCBFW-GJLSYRFBSA-N

Biochem/physiol Actions

Biphalin is a dimeric enkephalin that is a potent and non-selective opioid receptors (OR) agonist. It displays a high analgesic potency that is over 1000-fold greater than morphine. Studies show that biphalin exhibits neuroprotective effects in rat models of stroke.
Biphalin is a potent and non-selective opioid receptors (OR) agonist that displays neuroprotective effects in rat models of stroke.
Biphalin trifluoroacetate salt, a highly active synthetic octapeptide, is an analog of biphalin. It displays a strong affinity in the nanomolar range for the receptors μ and δ.

Features and Benefits

This compound is featured on the Opioid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

存储类别

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

历史批次信息供参考:

分析证书(COA)

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