Skip to Content
Merck
CN

SML3878

KMR-206

≥94% (HPLC)

Synonym(s):

6-(4-(2-fluoro-5-((4-oxo-7-(prop-1-yn-1-yl)-3,4-dihydrophthalazin-1-yl)methyl)benzoyl)piperazin-1-yl)nicotinonitrile

Sign In to View Organizational & Contract Pricing.

Select a Size


About This Item

Empirical Formula (Hill Notation):
C29H23FN6O2
CAS Number:
Molecular Weight:
506.53
NACRES:
NA.21
Assay:
≥94% (HPLC)
Form:
powder
Quality level:
Technical Service
Need help? Our team of experienced scientists is here for you.
Let Us Assist
Technical Service
Need help? Our team of experienced scientists is here for you.
Let Us Assist

SMILES string

O=C(C1=CC(CC2=NNC(C3=C2C=C(C=C3)C#CC)=O)=CC=C1F)N4CCN(CC4)C5=NC=C(C=C5)C#N

assay

≥94% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 2 mg/mL, clear

storage temp.

2-8°C

Quality Level

Biochem/physiol Actions

Cell penetrant, potent, and selective inhibitor of PARP7 that inhibits auto-MARylation and induced IFN-β in mouse colon carcinoma.
KMR-206 is a cell penetrant, potent, and selective inhibitor of PARP7 that inhibits auto-MARylation and induced IFN-β in mouse colon carcinoma (CT-26) cells. Also increased PARP7 protein levels in CT-26 cells.

Choose from one of the most recent versions:

Certificates of Analysis (COA)

Lot/Batch Number

Don't see the Right Version?

If you require a particular version, you can look up a specific certificate by the Lot or Batch number.

Already Own This Product?

Find documentation for the products that you have recently purchased in the Document Library.

Visit the Document Library

Z G Jia et al.
Zhonghua zhong liu za zhi [Chinese journal of oncology], 9(2), 124-126 (1987-03-01)
CT guided percutaneous fine needle aspiration cytodiagnosis was performed on 30 patients with pancreatic and periampullary tumors in China-Japan Friendship Hospital from November 1984 to January 1986. In our series, 9 pancreatic head cancers, 4 pancreatic body and tail cancers

Our team of scientists has experience in all areas of research including Life Science, Material Science, Chemical Synthesis, Chromatography, Analytical and many others.

Contact Technical Service