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Merck
CN

SML4092

SGC-GSK3-1

≥98% (HPLC)

Synonym(s):

4-(2,6-Difluorobenzamido)-N-((tetrahydro-2H-pyran-4-yl)methyl)-1H-pyrazole-3-carboxamide

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About This Item

Empirical Formula (Hill Notation):
C17H18F2N4O3
CAS Number:
Molecular Weight:
364.35
NACRES:
NA.28
Assay:
≥98% (HPLC)
Form:
powder
Quality level:
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SMILES string

O=C(NCC1CCOCC1)C2=NNC=C2NC(C3=C(C=CC=C3F)F)=O

assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 2 mg/mL, clear

storage temp.

2-8°C

Quality Level

Biochem/physiol Actions

Potent and selective glycogen synthase kinase-3 (GSK3⍺/β) inhibitor.

SGC-GSK3-1 is a potent and selective glycogen synthase kinase-3 inhibitor (GSK3⍺/β IC50 = 1/2 nM by cell-free enzymatic assay, 4.6/12 nM by cellular NanoBRET) that protects iPSC-derived motor neurons from ER stress-induced death.

Regulatory Information

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