119147
8-环戊基-1,3-二丙基黄嘌呤
DPCPX
别名:
1,3-二丙基-8-环戊基黄嘌呤, DPCPX, PD 116948
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关于此项目
经验公式（希尔记法）:
C16H24N4O2
化学文摘社编号:
分子量:
304.39
UNSPSC Code:
12352200
NACRES:
NA.51
MDL number:
产品名称
8-环戊基-1,3-二丙基黄嘌呤, DPCPX
InChI
1S/C16H24N4O2/c1-3-9-19-14-12(15(21)20(10-4-2)16(19)22)17-13(18-14)11-7-5-6-8-11/h11H,3-10H2,1-2H3,(H,17,18)
SMILES string
CCCN1C(=O)N(CCC)c2nc([nH]c2C1=O)C3CCCC3
InChI key
FFBDFADSZUINTG-UHFFFAOYSA-N
form
white solid
solubility
soluble (DMSO (5 mM))
storage temp.
2-8°C
Quality Level
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General description
A blood-brain barrier permeable xanthine derivative that acts as a highly selective antagonist of Adenosine A1 receptor (A1R; Ki = 3.9 nM, 130 nM, 1.0 µM, 4.0 µM for human A1, A2A, A2B, and A3 respectively). Exhibits about 1,000-fold higher affinity and a 30-fold greater selectivity for A1R when compared to theophylline. Shown to competitively antagonize the inhibition of adenylate cyclase activity via A1 adenosine receptors in rat fat cells and the stimulation of adenylate cyclase via A2 adenosine receptors in human platelets. Exhibits hypertensive properties.
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