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Merck
CN

370695

GW1929

PPARγ agonist, crystalline solid

别名:

GW1929, PPAR Agonist V, PPARγ Agonist IV

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关于此项目

经验公式（希尔记法）:
C30H29N3O4
化学文摘社编号:
196808-24-9
分子量:
495.57
MDL number:
MFCD04040003
UNSPSC Code:
12352200
NACRES:
NA.77
Form:
crystalline solid
Quality level:
100
Storage condition:
OK to freeze
protect from light

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产品名称

GW1929, A potent, tyrosine-based peroxisome proliferator-activated receptor γ (PPARγ) agonist (EC50 = 13 nM for murine receptor and 6.2 nM for human receptor in cell-based transactivation assays).

SMILES string

N([C@@H](Cc3ccc(cc3)OCCN(C)c4ncccc4)C(=O)O)c1c(cccc1)C(=O)c2ccccc2

InChI

1S/C30H29N3O4/c1-33(28-13-7-8-18-31-28)19-20-37-24-16-14-22(15-17-24)21-27(30(35)36)32-26-12-6-5-11-25(26)29(34)23-9-3-2-4-10-23/h2-18,27,32H,19-21H2,1H3,(H,35,36)/t27-/m0/s1

InChI key

QTQMRBZOBKYXCG-MHZLTWQESA-N

form

crystalline solid

manufacturer/tradename

Calbiochem®

storage condition

OK to freeze
protect from light

color

yellow

solubility

DMSO: 100 mg/mL

shipped in

ambient

storage temp.

−20°C

Quality Level

100

相关类别

Biochem/physiol Actions

Cell permeable: no
EC50 = 13 nM as peroxisome proliferator-activated receptor γ (PPARγ) agonist for murine receptor and 6.2 nM for human receptor in cell-based transactivation assays
Primary Target
Peroxisome proliferator-activated receptor γ (PPARγ) agonist
Product does not compete with ATP.
Reversible: no

Disclaimer

Toxicity: Standard Handling (A)

General description

A potent, tyrosine-based peroxisome proliferator-activated receptor γ (PPARγ) agonist (EC50 = 13 nM for murine PPARγ and 6.2 nM for human PPARγ in cell-based transactivation assays).

Other Notes

Han, S., et al. 2004. Clin. Cancer Res.10, 1911.
Willson, T.M., et al. 2000. J. Med. Chem.43, 527.
Brown, K.K., et al. 1999. Diabetes48, 1415.

Packaging

Packaged under inert gas

Preparation Note

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

存储类别

11 - Combustible Solids

wgk

WGK 1

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