form
solid
technique(s)
HPLC: suitable, gas chromatography (GC): suitable
color
pale yellow
solubility
ethanol: 11 mg/mL, 0.1 M HCl: 30 mg/mL, DMSO: 4.8 mg/mL
format
neat
SMILES string
CN1CCN(CC1)C2=Nc3cc(Cl)ccc3Nc4ccccc24
InChI
1S/C18H19ClN4/c1-22-8-10-23(11-9-22)18-14-4-2-3-5-15(14)20-16-7-6-13(19)12-17(16)21-18/h2-7,12,20H,8-11H2,1H3
InChI key
QZUDBNBUXVUHMW-UHFFFAOYSA-N
Gene Information
human ... DRD2(1813), HTR2A(3356)
Application
Refer to the product′s Certificate of Analysis for more information on a suitable instrument technique. Contact Technical Service for further support.
Biochem/physiol Actions
非典型抗精神病药，对 D4 多巴胺受体比对 D2 或 D3 多巴胺受体表现出更大的亲和性；在用典型抗精神病药无效的患者中，对精神分裂症的阳性和阴性症状均表现出抗精神病疗效。
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