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D8040

反式 -U-50488 甲磺酸盐

Name: 反式 </I>-U-50488 甲磺酸盐
Brand: SIGMA

别名:

反 -(±)-3,4-二氯-N-甲基-N- [2-（1-吡咯烷基）环己基] 苯乙酰胺甲磺酸盐, U-50488H

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关于此项目

经验公式（希尔记法）:

C₁₉H₂₆Cl₂N₂O · CH₄O₃S

分子量:

465.43

NACRES:

NA.77

PubChem Substance ID:

24278070

UNSPSC Code:

12352106

MDL number:

MFCD00133867

Form:

powder

Quality level:

200

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form

powder

Quality Level

200

solubility

H₂O: 50 mg/mL

storage temp.

2-8°C

SMILES string

CS(O)(=O)=O.CN([C@@H]1CCCC[C@H]1N2CCCC2)C(=O)Cc3ccc(Cl)c(Cl)c3

InChI

1S/C19H26Cl2N2O.CH4O3S/c1-22(19(24)13-14-8-9-15(20)16(21)12-14)17-6-2-3-7-18(17)23-10-4-5-11-23;1-5(2,3)4/h8-9,12,17-18H,2-7,10-11,13H2,1H3;1H3,(H,2,3,4)/t17-,18-;/m1./s1

InChI key

OJPHNZCUXUUVKU-JAXOOIEVSA-N

Gene Information

human ... OPRK1(4986)

Application

(±)-反式-U-50488 甲磺酸盐已被用作 κ -阿片受体的对照激动剂。

Biochem/physiol Actions

选择性 κ-已知阿片受体激动剂 (±)-反式-U-50488 甲磺酸盐可诱导利尿。研究发现 U-50488H 与其联合给药时可预防吗啡耐受。

存储类别

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)

历史批次信息供参考:

分析证书(COA)

Lot/Batch Number

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全球贸易项目编号

货号	GTIN
D8040-100MG	04061833589151
D8040-50MG	04061832862101
D8040-10MG	04061832862095

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