E1905
(+)-依托莫西 钠盐 水合物
≥98% (HPLC), powder, CPT-1 inhibitor
别名:
R(+)-2-[6-(4-氯苯氧基）己基]-环氧乙烷-2-羧酸 钠盐 水合物
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关于此项目
经验公式（希尔记法）:
C15H18ClO4 · Na · H2O
化学文摘社编号:
分子量:
338.76
MDL编号:
UNSPSC代码:
12352200
PubChem化学物质编号:
NACRES:
NA.77
产品名称
(+)-依托莫西 钠盐 水合物, ≥98% (HPLC), powder
质量水平
方案
≥98% (HPLC)
表单
powder
颜色
white
溶解性
H2O: freely soluble
储存温度
2-8°C
SMILES字符串
O.[Na+].[O-]C(=O)[C@@]2(CCCCCCOc1ccc(Cl)cc1)CO2
InChI
1S/C15H19ClO4.Na.H2O/c16-12-5-7-13(8-6-12)19-10-4-2-1-3-9-15(11-20-15)14(17)18;;/h5-8H,1-4,9-11H2,(H,17,18);;1H2/q;+1;/p-1/t15-;;/m1../s1
InChI key
WENJLJJSJDAJDN-QCUBGVIVSA-M
一般描述
(+)-依托莫西钠盐水合物属于环氧乙烷羧酸基团化合物，调节脂肪酸前体代谢通道。它有利于T细胞氧化压力并且防止T细胞分化。它能抑制脂肪酸代谢，促使饥饿和食物摄入。依托莫西削弱髓源抑制性细胞介导的肿瘤，可能具有治疗潜在价值。
应用
(+)-依托莫西钠盐水合物可用作乳腺肿瘤细胞系和小鼠肿瘤肉毒碱棕榈酰转移酶1（CTP-1）的抑制剂。它还可以用于人原发性前列腺上皮细胞和淋巴细胞的脂肪酸氧化抑制物。
生化/生理作用
不可逆O—肉毒碱棕榈酰转移酶1（CTP-1）抑制剂；PPARα 激活剂
包装
气密保存，隔绝光照
警示用语：
Danger
危险声明
危险分类
Acute Tox. 3 Oral
储存分类代码
6.1C - Combustible acute toxic Cat.3 / toxic compounds or compounds which causing chronic effects
WGK
WGK 3
闪点(°F)
Not applicable
闪点(°C)
Not applicable
个人防护装备
dust mask type N95 (US), Eyeshields, Faceshields, Gloves
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