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Merck
CN

G7791

GW8510

solid

别名:

4-{[(7-Oxo-6,7-dihydro-8H-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}-N-(2-pyridyl)benzenesulfonamide

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选择尺寸


关于此项目

经验公式(希尔记法):
C21H15N5O3S2
化学文摘社编号:
分子量:
449.51
NACRES:
NA.77
PubChem Substance ID:
UNSPSC Code:
12352202
MDL number:
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产品名称

GW8510, solid

InChI

1S/C21H15N5O3S2/c27-21-15(19-16(25-21)8-9-17-20(19)30-12-24-17)11-23-13-4-6-14(7-5-13)31(28,29)26-18-3-1-2-10-22-18/h1-12,23H,(H,22,26)(H,25,27)/b15-11-

SMILES string

O=C1Nc2ccc3ncsc3c2\C1=C\Nc4ccc(cc4)S(=O)(=O)Nc5ccccn5

InChI key

GCYXEGSPUDSZJY-PTNGSMBKSA-N

assay

~98% (HPLC)

form

solid

solubility

DMSO: soluble

storage temp.

room temp

Quality Level

Gene Information

human ... CDC2(983), CDK2(1017)

Biochem/physiol Actions

最初作为细胞周期蛋白依赖性激酶 2(CDK2)的抑制剂,随后的研究表明 GW8510 是非选择性的。

Legal Information

根据葛兰素史克的协议出售,用于研究目的

存储类别

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)


历史批次信息供参考:

分析证书(COA)

Lot/Batch Number

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