R123
RBI 257 maleate salt
solid
别名:
1-[4-Iodobenzyl]-4-[[2-[3-isopropoxy]pyridyl]-methylamino]piperidine maleate salt, p-Iodo-U-101,958 maleate salt
表单
solid
颜色
white
溶解性
H2O: 0.2 mg/mL
ethanol: 1 mg/mL
0.1 M HCl: 7 mg/mL
DMSO: 9 mg/mL
储存温度
2-8°C
SMILES字符串
[H]\C(=C(/[H])C(O)=O)C(O)=O.CC(C)Oc1cccnc1N(C)C2CCN(CC2)Cc3ccc(I)cc3
生化/生理作用
High affinity D4 dopamine receptor ligand.
储存分类代码
13 - Non Combustible Solids
WGK
WGK 3
闪点(°F)
Not applicable
闪点(°C)
Not applicable
个人防护装备
Eyeshields, Gloves, type N95 (US)
法规信息
新产品
此项目有
N S Kula et al.
European journal of pharmacology, 331(2-3), 333-336 (1997-07-23)
RBI-257 (1-[4-iodobenzyl]-4-[N-(3-isopropoxy-2-pyridinyl)-N-methyl]-aminopiperid ine), the p-iodobenzyl analog of U-101,958 (1-benzyl-4-[N-(3-isopropoxy-2-pyridinyl)-N-methyl]-aminopiperidine) had a lower dissociation constant (Ki = 0.3 vs. 2.7 nM) and higher selectivity than U-101,958 at dopamine D4 receptors, over dopamine D2 and D3 receptors in transfected cell membranes and
Compounds selective for dopamine receptor subtypes.
Kebabian, et al.
Drug Discovery Today, 2, 333-340 (1997)
F Henry et al.
Theriogenology, 83(8), 1373-1380 (2015-03-05)
From many endangered or threatened species which are expected to profit from assisted reproduction techniques, mainly epididymal sperm of dead or freshly castrated males are available. These sperm had contact to epididymal secretion products but not to seminal fluid components.
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