S106
SR-95531
≥98% (HPLC), GABAA receptor antagonist , powder
别名:
2-（3-羧丙基）-3-氨基-6-（4-甲氧基苯基）哒嗪溴化物, 加巴嗪
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关于此项目
经验公式（希尔记法）:
C15H18BrN3O3
化学文摘社编号:
分子量:
368.23
UNSPSC Code:
12352200
PubChem Substance ID:
NACRES:
NA.77
MDL number:
产品名称
SR-95531, ≥98% (HPLC), powder
SMILES string
[Br-].COc1ccc(cc1)-c2ccc(N)[n+](CCCC(O)=O)n2
InChI key
GFZHNFOGCMEYTA-UHFFFAOYSA-N
InChI
1S/C15H17N3O3.BrH/c1-21-12-6-4-11(5-7-12)13-8-9-14(16)18(17-13)10-2-3-15(19)20;/h4-9,16H,2-3,10H2,1H3,(H,19,20);1H
assay
≥98% (HPLC)
form
powder
color
white
solubility
H2O: >10 mg/mL
Quality Level
Gene Information
human ... GABRA1(2554), GABRA2(2555), GABRA3(2556), GABRA4(2557), GABRA5(2558), GABRA6(2559), GABRB1(2560), GABRB2(2561), GABRB3(2562)
rat ... Gabra2(29706)
相关类别
Biochem/physiol Actions
SR-95531 是一种特异性 GABA a 受体拮抗剂，不影响 GABA 转氨酶或谷氨酸脱羧酶活性。
Features and Benefits
这种化合物是神经科学研究的特色产品。点击此处发现更多特色神经科学产品。在sigma.com/discover-bsm可了解更多关于生物活性小分子的其他研究领域。
存储类别
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
ppe
Eyeshields, Gloves, type N95 (US)
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