SML0936
特立氟胺
≥98% (HPLC), anti-inflammatory immunomodulator, powder
别名:
(Z)-2-氰基-3-羟基-N- [4-（三氟甲基）苯基]-2-丁烯酰胺, A 1726, A77-1726, A771726, HMR 1726, N-（4-三氟甲基苯基）-2-氰基-3-羟基克罗胺, SU 20, 氟酰胺
产品名称
特立氟胺, ≥98% (HPLC)
InChI
1S/C12H9F3N2O2/c1-7(18)10(6-16)11(19)17-9-4-2-8(3-5-9)12(13,14)15/h2-5,18H,1H3,(H,17,19)/b10-7-
InChI key
UTNUDOFZCWSZMS-YFHOEESVSA-N
assay
≥98% (HPLC)
form
powder
color
white to beige
solubility
DMSO: 5 mg/mL, clear (warmed)
storage temp.
−20°C
Quality Level
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相关类别
Application
特立氟胺是一种二氢乳清酸脱氢酶 (DHODH) 抑制剂。
Biochem/physiol Actions
特立氟胺是一种可口服的抗炎免疫调节剂。
特立氟胺是一种可口服的抗炎免疫调节剂。阻断二氢乳清酸脱氢酶的活性，阻止嘧啶合成及 T、B 细胞增殖和功能。特立氟胺用于治疗风湿性关节炎，最近被批准用于多发性硬化症。
signalword
Warning
hcodes
Hazard Classifications
Acute Tox. 4 Oral
存储类别
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
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商品
Bioactive small molecules for immune system signaling target identification/validation and antibiotics, antivirals, and antifungals offered.
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