Quality Segment
assay
≥98% (HPLC)
form
powder
color
white to beige
solubility
0.2 mg/mL (DMSO:EtOH (2:1),clear, warmed, clear colorless solution)
storage temp.
room temp
SMILES string
[o]1c2c([c](cc1c3cc(ccc3)O)=O)c(ccc2)O
InChI key
SZMQXDYEGKRZDG-UHFFFAOYSA-N
Biochem/physiol Actions
Cell penetrant, selective and potent inhibitor of the androgen receptor (AR)-ELK1 interaction
KCI807 is a cell penetrant, selective and potent inhibitor of the androgen receptor (AR)-ELK1 interaction. KCI807 interrupts association of the androgen receptor (AR) with transcription activator ELK1 (ETS family transcription factor ELK1). It potently suppresses growth of enzalutamide-resistant prostate cancer tumor xenografts in rodents.
存储类别
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable