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关于此项目
经验公式（希尔记法）:
C14H13N3OS3
化学文摘社编号:
分子量:
335.47
MDL number:
NACRES:
NA.21
UNSPSC Code:
12352200
eCl@ss:
32160703
Assay:
≥98% (HPLC)
Form:
powder
Quality Segment
assay
≥98% (HPLC)
form
powder
color
white to beige
solubility
DMSO: 2 mg/mL, clear
storage temp.
2-8°C
SMILES string
CC1=C(CNC(NC2=CC=CS2)=O)SC(C3=CC=CS3)=N1
Biochem/physiol Actions
Potent and highly selective inhibitor of vascular Kir6.1/SUR2B (vascular KATP) channels.
VU0542270 is a potent and highly selective inhibitor of vascular Kir6.1/SUR2B (vascular KATP) channels (IC50 ~ 100 nM) that show no apparent activity toward Kir6.2/SUR1 and other members of the Kir channel family. It appears that VU0542270 binds to SUR2. It has a rather short in vivo half-life (t1/2 = 0.64 hour).
VU0542270 is a potent and highly selective inhibitor of vascular Kir6.1/SUR2B (vascular KATP) channels (IC50 ~ 100 nM) that show no apparent activity toward Kir6.2/SUR1 and other members of the Kir channel family. It appears that VU0542270 binds to SUR2. It has a rather short in vivo half-life (t1/2 = 0.64 hour).
存储类别
11 - Combustible Solids
WGK
WGK 3
闪点 (F)
Not applicable
闪点 (°C)
Not applicable