SML4111

Gepirone hydrochloride

Name: Gepirone hydrochloride
Brand: SIGMA

≥98% (HPLC)

别名:

4,4-Dimethyl-1-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-2,6-piperidinedione hydrochloride, 4,4-dimethyl-1-(4-(4-(pyrimidin-2-yl)piperazin-1-yl)butyl)piperidine-2,6-dione hydrochloride, BMY 13805, BMY 13805-1, ORG-13011

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关于此项目

经验公式（希尔记法）:

C₁₉H₂₉N₅O₂ · xHCl

化学文摘社编号:

108964-56-3

分子量:

359.47 (free base basis)

MDL number:

MFCD00868196

NACRES:

NA.28

Assay:

≥98% (HPLC)

Form:

powder

Quality level:

100

Storage condition:

desiccated

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SMILES string

O=C1N(C(CC(C1)(C)C)=O)CCCCN2CCN(C3=NC=CC=N3)CC2.[xHCl]

assay

≥98% (HPLC)

form

powder

storage condition

desiccated

color

white to beige

solubility

H₂O: 2 mg/mL, clear

storage temp.

-10 to -25°C

Quality Level

100

Biochem/physiol Actions

Orally bioavailable, potent, and selective partial agonist of serotonin 5-HT1A receptor; non-sedative anxiolytic and antidepressant drug.
Gepirone hydrochloride is an orally bioavailable, non-sedative anxiolytic and antidepressant drug of the buspirone family with a unique mechanism of action that differs from other antidepressants and anxiolytic drugs. Gepirone acts as a partial serotonin 5-HT1A receptor agonist with differential action at pre-and postsynaptic 5-HT1A receptors. Gepirone is much more efficacious than selective serotonin reuptake inhibitors (SSRIs) without causing sexual dysfunction.