SML4120
BIBP3226 trifluoroacetate
≥95% (HPLC)
别名:
BIBP 3226 TFA salt, BIBP-3226 TFA salt, Diphenylacetyl-D-Arg-4-hydroxybenzylamide, trifluoroacetate salt, N2-(Diphenylacetyl)-N-[(4-hydroxyphenyl)methyl]-D-arginine amide, trifluoroacetate salt, (R)-N2-(Diphenylacetyl)-N-[(4-hydroxyphenyl)methyl]-argininamide, trifluoroacetate salt
质量水平
方案
≥95% (HPLC)
表单
powder
储存条件
desiccated
颜色
white to beige
溶解性
DMSO: 2 mg/mL, clear
储存温度
2-8°C
SMILES字符串
OC(C=C1)=CC=C1CNC([C@@H](CCCNC(N)=N)NC(C(C2=CC=CC=C2)C3=CC=CC=C3)=O)=O
生化/生理作用
Potent and selective non-peptide neuropeptide Y receptor Y1 antagonist in vitro and in vivo.
BIBP3226 is a potent and selective non-peptide neuropeptide Y receptor Y1 antagonist (Ki = 7 nM against neuropeptide Y binding to receptor Y1) in vitro and in vivo. BIBP3226 selectively blocks Y1 receptor-mediated rabbit saphenous vein contraction (pA2 = 7.36), but not receptor Y2- or Y3-dependent biological effects.
BIBP3226 is a potent and selective non-peptide neuropeptide Y receptor Y1 antagonist (Ki = 7 nM against neuropeptide Y binding to receptor Y1) in vitro and in vivo. BIBP3226 selectively blocks Y1 receptor-mediated rabbit saphenous vein contraction (pA2 = 7.36), but not receptor Y2- or Y3-dependent biological effects.
免责声明
Hygroscopic
法规信息
新产品
此项目有
历史批次信息供参考:
分析证书(COA)
Lot/Batch Number
我们的科学家团队拥有各种研究领域经验，包括生命科学、材料科学、化学合成、色谱、分析及许多其他领域.
联系客户支持