SML4120

BIBP3226 trifluoroacetate

Name: BIBP3226 trifluoroacetate
Brand: SIGMA

≥95% (HPLC)

别名:

BIBP 3226 TFA salt, BIBP-3226 TFA salt, Diphenylacetyl-D-Arg-4-hydroxybenzylamide, trifluoroacetate salt, N2-(Diphenylacetyl)-N-[(4-hydroxyphenyl)methyl]-D-arginine amide, trifluoroacetate salt, (R)-N2-(Diphenylacetyl)-N-[(4-hydroxyphenyl)methyl]-argininamide, trifluoroacetate salt

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关于此项目

经验公式（希尔记法）:

C₂₇H₃₁N₅O₃ · xC₂HF₃O₂

化学文摘社编号:

1068148-47-9

分子量:

473.57 (free base basis)

MDL number:

MFCD00938562

NACRES:

NA.28

Assay:

≥95% (HPLC)

Form:

powder

Quality level:

100

Storage condition:

desiccated

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SMILES string

OC(C=C1)=CC=C1CNC([C@@H](CCCNC(N)=N)NC(C(C2=CC=CC=C2)C3=CC=CC=C3)=O)=O

assay

≥95% (HPLC)

form

powder

storage condition

desiccated

color

white to beige

solubility

DMSO: 2 mg/mL, clear

storage temp.

2-8°C

Quality Level

100

Biochem/physiol Actions

Potent and selective non-peptide neuropeptide Y receptor Y1 antagonist in vitro and in vivo.
BIBP3226 is a potent and selective non-peptide neuropeptide Y receptor Y1 antagonist (Ki = 7 nM against neuropeptide Y binding to receptor Y1) in vitro and in vivo. BIBP3226 selectively blocks Y1 receptor-mediated rabbit saphenous vein contraction (pA2 = 7.36), but not receptor Y2- or Y3-dependent biological effects.