Quality Segment
assay
≥98% (HPLC)
form
powder
color
white to beige
solubility
DMSO: 2 mg/mL, clear
storage temp.
-10 to -25°C
Biochem/physiol Actions
Apatinib (rivoceranib) is an orally available, potent, and selective inhibitor of vascular endothelial growth factor receptor 2 (VEGFR2) (IC50 = 1 nM) that potently blocks tumor angiogenesis and inhibits tumor growth. Apatinib exhibits encouraging antitumor efficacy and acceptable toxicities in multiple clinical trials. It also mildly targets c-Kit and c-SRC tyrosine kinases.
警示词
Warning
危险代码
Hazard Classifications
Acute Tox. 4 Oral
存储类别
11 - Combustible Solids
闪点 (F)
Not applicable
闪点 (°C)
Not applicable