U101
5-Methylurapidil
solid
别名:
5-Methyl-6[[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]amino]-1,3-dimethyluracil
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关于此项目
经验公式（希尔记法）:
C21H31N5O3
化学文摘社编号:
分子量:
401.50
NACRES:
NA.77
PubChem Substance ID:
UNSPSC Code:
12352200
MDL number:
Form:
solid
form
solid
Quality Segment
color
white
solubility
H2O: 0.4 mg/mL, 0.1 M HCl: 3.8 mg/mL
SMILES string
Cl[H].COc1ccccc1N2CCN(CCCNC3=C(C)C(=O)N(C)C(=O)N3C)CC2
InChI
1S/C21H31N5O3.ClH/c1-16-19(23(2)21(28)24(3)20(16)27)22-10-7-11-25-12-14-26(15-13-25)17-8-5-6-9-18(17)29-4;/h5-6,8-9,22H,7,10-15H2,1-4H3;1H
InChI key
WAZDYFHTLYHMKO-UHFFFAOYSA-N
Gene Information
human ... ADRA1A(148), ADRA1B(147), ADRA1D(146)
Application
5-Methylurapidil has been used for competitive binding in radioligand binding assays.
Biochem/physiol Actions
Selective α1A-adrenoceptor antagonist; antihypertensive.
Features and Benefits
This compound is featured on the α1-Adrenoceptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
Preparation Note
5-Methylurapidil is soluble in water at 0.4 mg/ml and is also soluble in 0.1 M HCl at 3.8 mg/ml.
存储类别
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
ppe
Eyeshields, Gloves, type N95 (US)
商品
Review alpha 1 adrenoceptors as well as their agonists, antagonists, and tissue expression patterns. We suggest several modulators and alternatives for working with a-1 adrenoreceptors.
相关内容
Instructions
全球贸易项目编号
| 货号 | GTIN |
|---|---|
| EPP0625-0020-1EA | 04061835083091 |
| U101-50MG | 04061832094151 |
| U101-10MG | 04061832094144 |