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SML2173

NS3861

≥98% (HPLC)

Synonym(s):

3-(3-Bromo-2-thienyl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene, NS 3861

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About This Item

Empirical Formula (Hill Notation):
C12H14BrNS
CAS Number:
216853-59-7
Molecular Weight:
284.22
UNSPSC Code:
12352200
NACRES:
NA.77
Assay:
≥98% (HPLC)
Form:
powder
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assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 2 mg/mL, clear

storage temp.

2-8°C

SMILES string

BrC1=C(SC=C1)C2=CC(N3C)CCC3C2

InChI key

ZJCNRVHZJADROC-UHFFFAOYSA-N

Biochem/physiol Actions

α3β2 heteromeric neuronal nAChRs agonist
NS3861 is a neuronal nicotinic receptor agonist that selectively activates α3 containing nAChRs and it displays higher efficacy at the α3β2 receptor compared with the α3β4 receptor. NS3861 does not activate α4 containing receptors. NS3861 was reported to reverse chronic opioid-induced constipation in vivo.

Storage Class

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

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