513210

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Showing 1-7 of 7 results for "513210" within Papers

Synthesis and structure-activity relationships of novel benzofuran farnesyltransferase inhibitors.

Asoh K, et al.

Bioorganic & Medicinal Chemistry Letters, 19(6), 1753-1757 (2009)

20-Aminosteroids as a novel class of selective and complete androgen receptor antagonists and inhibitors of prostate cancer cell growth.

Fousteris MA, et al.

Bioorganic & Medicinal Chemistry Letters, 18(19), 6960-6969 (2010)

Highly stereoselective addition of organometallic reagents to N-tert-butanesulfinyl imines derived from 3- and 4-substituted cyclohexanones.

Jeffrey P McMahon et al.

Organic letters, 6(10), 1645-1647 (2004-05-07)

Addition of alkyl or aryl Grignard reagents to N-sulfinyl imines derived from 3- and 4-substituted cyclohexanones proceeds with good yields and with excellent diasteroselectivity. The selectivity of the reaction is controlled by the ring substituent rather than the sulfinyl group

Asymmetric syntheses of 1-aryl-2,2,2-trifluoroethylamines via diastereoselective 1,2-addition of arylmetals to 2-methyl-N-(2,2,2-trifluoroethylidene)propane-2-sulfinamide.

Vouy Linh Truong et al.

Organic letters, 9(4), 683-685 (2007-01-30)

Condensation of N-tert-butanesulfinamide (S)-1 with trifluoroacetaldehyde hydrate 2a afforded 2-methyl-N-(2,2,2-trifluoroethylidene)propane-2-sulfinamide 3. Without isolation and purification, imine 3 was added to various aryllithium reagents to give highly diastereomerically enriched adducts 5a-g. Acidic methanolysis of 5a-g provided the desired 1-aryl-2,2,2-trifluoroethylamine hydrochloride compounds

Journal of the American Chemical Society, 119, 9913-9914 (1997)

N-tert-butanesulfinyl imines: versatile intermediates for the asymmetric synthesis of amines.

Jonathan A Ellman et al.

Accounts of chemical research, 35(11), 984-995 (2002-11-20)

N-tert-Butanesulfinyl aldimines 3 and ketimines 4 are exceedingly versatile intermediates for the asymmetric synthesis of amines. The N-tert-butanesulfinyl imines are prepared in high yields by condensing enantiomerically pure tert-butanesulfinamide 1, which is readily available in either configuration, with a wide

Organic Letters, 69, 1800-1800 (2004)

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