326 HDAC-3 H3034 8841 HDAC3 P NP_003874.2 y y y
316 hABH1 A8103 8846 ALKBH1 M NP_006011.2 y n/d n/d
531 p300/CBP P2859 8850 KAT2B M NP_003875.3 y y y
557 PCAF P7493 8850 KAT2B P NP_003875.3 y n/d n/d
533
326 HDAC-3 H3034 8841 HDAC3 P NP_003874.2 y y y
316 hABH1 A8103 8846 ALKBH1 M NP_006011.2 y n/d n/d
531 p300/CBP P2859 8850 KAT2B M NP_003875.3 y y y
557 PCAF P7493 8850 KAT2B P NP_003875.3 y n/d n/d
533
326 HDAC-3 H3034 8841 HDAC3 P NP_003874.2 y y y
316 hABH1 A8103 8846 ALKBH1 M NP_006011.2 y n/d n/d
531 p300/CBP P2859 8850 KAT2B M NP_003875.3 y y y
557 PCAF P7493 8850 KAT2B P NP_003875.3 y n/d n/d
533
-668 3
DYRK1A, active 14-435
DYRK2, active 14-669 3
eEF-2K, active 14-654 3 12-550
EGFR, active 14-531 3
EGFR (L858R), active 14-626 3
EGFR (L861Q), active 14-627 3
EGFR (T790M), active 14-725 3
EGFR (T790M
Butyl-4-(2-chlorophenyl)-9-hydroxypyrrolo[3,4-c]carbazole-1,3-(2h,6h)-dione}
A pyrrolocarbazole compound that acts as a potent, ATP-binding site-
targeting inhibitor of Wee1 (IC50 = 59 nM) with a ~590-fold
.1 M y n/d n/d
530 p21WAF1/Cip1 P1484 12575, 1026 CDKN1A,Cdkn1a NP_031695.1,NP_510867.1 M y y n/d
531 p300/CBP P2859 18519, 8850, 301164 Pcaf,PCAF NP_064389.2,NP_003875.3,NP_001019423.1 M y y y
532 p34cdc2
528 Anti Cy3+Cy5 C0992 M NA NA NA
529 p19INK4d P4354 M y n/d n/d
530 p21WAF1/Cip1 P1484 M y y n/d
531 p300/CBP P2859 M y y y
532 p34cdc2 C3085 M y y n/d
533 p35 (Cdk5 Regulator) P9489 P y
Alexa Fluor 555 9H2 H M FC IF M IgG1κ 25 µg 16-245
Conjugate
Kinase
EGFR, active 10 µg 14-531
EGFR (L858R), active 10 µg 14-626
EGFR (L861Q), active 10 µg 14-627
EGFR (T790M)
function, stopwatch, loud alert sound.
Time indication is switchable from
999 min., 59 sec. to 9 h, 59 min., 59
sec., 1/10 sec..
Incl. battery (AA)
Colour: pigeon blue
Dimensions: 170 x 130 x 80