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Merck
CN

SML0424

ST247

≥98% (HPLC)

别名:

3-[[[4-(Hexylamino)-2-methoxyphenyl]amino]sulfonyl]-2-thiophenecarboxylic acid methyl ester

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关于此项目

经验公式（希尔记法）:
C19H26N2O5S2
化学文摘社编号:
1356497-91-0
分子量:
426.55
UNSPSC Code:
12352200
PubChem Substance ID:
329825419
NACRES:
NA.77

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SMILES string

CCCCCCNc1ccc(NS(=O)(=O)c2ccsc2C(=O)OC)c(OC)c1

InChI

1S/C19H26N2O5S2/c1-4-5-6-7-11-20-14-8-9-15(16(13-14)25-2)21-28(23,24)17-10-12-27-18(17)19(22)26-3/h8-10,12-13,20-21H,4-7,11H2,1-3H3

InChI key

MRWCGEOYGFZZCJ-UHFFFAOYSA-N

assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 10 mg/mL (clear solution)

storage temp.

2-8°C

Quality Level

100

相关类别

Biochem/physiol Actions

ST247 is a PPAR β/δ inverse agonist.
ST247 is a PPAR β/δ selective inverse agonist. The compound is based on the structure of GSK0660, and is 10-fold more potent in blocking the transcription of endogenous target genes: ST247 IC50 = 19 nm vs. GSK0660 IC50 = 210 nM.

存储类别

11 - Combustible Solids

wgk

WGK 3

法规信息

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分析证书(COA)

Lot/Batch Number
0000060369
082M4602V

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