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Merck
CN

P5015

Sigma-Aldrich

Protein Kinase Inhibitor from rabbit muscle

lyophilized powder, 0.2-1 inhibitor U/μg protein

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About This Item

MDL number:
UNSPSC Code:
12352202
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biological source

rabbit muscle

form

lyophilized powder

specific activity

0.2-1 inhibitor U/μg protein

composition

Protein, ~95% biuret

storage temp.

2-8°C

Biochem/physiol Actions

Binds to the catalytic subunit of cyclic-AMP dependent protein kinase, displacing the regulatory subunit and inhibiting phosphorylating activity. The cAMP binding capacity of the regulatory subunit is enhanced. The amino acid sequence deduced from cDNA is 100% homologous with human PKI.

Packaging

Package size based on protein content.

Physical form

Lyophilized powder containing 5% potassium phosphate buffer salts

Preparation Note

Fractionated essentially by procedure of Walsh, D.A., et al., J. Biol. Chem., 246, 1977 (1971), through TCA precipitation.

Analysis Note

Crude

Other Notes

One unit will transfer 1.0 picomole (10-12 mol) of phosphate from γ-32P-ATP to hydrolyzed and partially dephosphorylated casein (Product No. C 4765) per min at pH 6.5 at 30 °C.

Storage Class Code

13 - Non Combustible Solids

WGK

WGK 3

Flash Point(F)

Not applicable

Flash Point(C)

Not applicable

Personal Protective Equipment

dust mask type N95 (US), Eyeshields, Gloves

Regulatory Information

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J Stern et al.
The Journal of general physiology, 85(2), 157-169 (1985-02-01)
The effect of intracellular nucleotides on the rate of spontaneous quantum bumps in Limulus ventral photoreceptors has been examined. Internal dialysis of photoreceptors with solutions lacking nucleotide leads to an elevation of the quantum bump rate that can be reversed
R O Arellano et al.
Biophysical journal, 57(2), 363-367 (1990-02-01)
The regulation of the cell-to-cell pathway formed by gap junctions seems to involve the interaction of the junctional channels with either calcium or hydrogen ions, as well as protein phosphorylation and calmodulin. These mechanisms of junctional regulation have been considered

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