PZ0112
PD-184161
≥98% (HPLC)
Synonym(s):
5-Bromo-2-[(2-chloro-4-iodophenyl)amino]-N-(cyclopropylmethoxy)-3,4-difluoro-benzamide, PF-1529483, PF-3011370, UK-287074
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About This Item
Empirical Formula (Hill Notation):
C17H13BrClF2IN2O2
CAS Number:
Molecular Weight:
557.56
NACRES:
NA.77
PubChem Substance ID:
UNSPSC Code:
12352200
MDL number:
Quality Level
assay
≥98% (HPLC)
form
powder
color
white to off-white
solubility
DMSO: >10 mg/mL
storage temp.
2-8°C
SMILES string
Fc1c(F)c(Nc2ccc(I)cc2Cl)c(cc1Br)C(=O)NOCC3CC3
InChI
1S/C17H13BrClF2IN2O2/c18-11-6-10(17(25)24-26-7-8-1-2-8)16(15(21)14(11)20)23-13-4-3-9(22)5-12(13)19/h3-6,8,23H,1-2,7H2,(H,24,25)
InChI key
VJNZMSLGVUSPCF-UHFFFAOYSA-N
Biochem/physiol Actions
PD-184161 is a MEK inhibitor.
Features and Benefits
This compound is featured on the MAPKKKs page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
Storage Class
11 - Combustible Solids
flash_point_f
Not applicable
flash_point_c
Not applicable
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Global Trade Item Number
| SKU | GTIN |
|---|---|
| PZ0112-25MG | 04061832449135 |
| PZ0112-5MG | 04061832449142 |