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SML3637

YM-254890

Name: YM-254890
Brand: SIGMA

≥95% (HPLC), Gαq/11 protein inhibitor, Powder or Lyophilized powder or film

Synonym(s):

N-Acetyl-L-threonyl-(aR)-a-hydroxybenzenepropanoyl-2,3-didehydro-N-methylalanyl-L-alanyl-N-methyl-L-alanyl-(3R)-3-[[(2S,3R)-2-(acetylamino)-3-hydroxy-4-methyl-1-oxopentyl]oxy]-L-leucyl-N,O-dimethyl-L-threonine (7→1)-lactone, QS 3666A, YM 254890

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About This Item

Empirical Formula (Hill Notation):

C₄₆H₆₉N₇O₁₅

CAS Number:

568580-02-9

Molecular Weight:

960.08

UNSPSC Code:

12352200

NACRES:

NA.77

MDL number:

MFCD09832722

Assay:

≥95% (HPLC)

Form:

(Powder or Lyophilized powder or film)

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Properties

Product Name

YM-254890, ≥95% (HPLC)

Quality Segment

100

assay

≥95% (HPLC)

form

(Powder or Lyophilized powder or film)

color

white to off-white

storage temp.

-10 to -25°C

Description

Biochem/physiol Actions

Gaq/11 protein inhibitor

YM-254890, a cyclic depsipeptide isolated from the culture broth of Chromobacterium sp., is a cell-permeable, potent and selective inhibitor of Gαq/11 protein. YM-254890 specifically inhibits the GDP/GTP exchange by blocking GDP release from the Gq protein.

Storage Class

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

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