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Merck
CN

T5830

Trap-101 hydrochloride

≥98% (HPLC), powder

Synonym(s):

1-[1-(cyclooctylmethyl)-1,2,3,6-tetrahydro-5-(hydroxymethyl)-4-pyridinyl]-3-ethyl-1,3-dihydro-2Hbenzimidazol-2-one hydrochloride

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About This Item

Empirical Formula (Hill Notation):
C24H35N3O2·HCl
CAS Number:
1216621-00-9
Molecular Weight:
434.01
NACRES:
NA.77
PubChem Substance ID:
329826831
UNSPSC Code:
12352200
MDL number:
MFCD09971083

Key Documents

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InChI key

YEVMLMQAMCKVSC-UHFFFAOYSA-N

SMILES string

Cl.CCN1C(=O)N(C2=C(CO)CN(CC2)CC3CCCCCCC3)c4ccccc14

InChI

1S/C24H35N3O2.ClH/c1-2-26-22-12-8-9-13-23(22)27(24(26)29)21-14-15-25(17-20(21)18-28)16-19-10-6-4-3-5-7-11-19;/h8-9,12-13,19,28H,2-7,10-11,14-18H2,1H3;1H

assay

≥98% (HPLC)

form

powder

color

white to off-white

solubility

H2O: ≥10 mg/mL

storage temp.

2-8°C

Biochem/physiol Actions

Trap-101 Hydrochloride is a nociceptin/orphanin FQ peptide (NOP) receptor blocker.
Trap-101 Hydrochloride is a nociceptin/orphanin FQ peptide (NOP) receptor blocker. Trap-101 acts as an inverse agonist. Trap-101 had been found to be an effective NOP receptor antagonist both in vitro and in vivo, with equivalent potency to J113397.

pictograms

Skull and crossbones
GHS06

signalword

Danger

hcodes

H301

Hazard Classifications

Acute Tox. 3 Oral

Storage Class

6.1C - Combustible acute toxic Cat.3 / toxic compounds or compounds which causing chronic effects

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

Regulatory Information

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Certificates of Analysis (COA)

Lot/Batch Number
100M4629V

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