Key Documents

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U101

5-Methylurapidil

Name: 5-Methylurapidil
Brand: SIGMA

solid

Synonym(s):

5-Methyl-6[[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]amino]-1,3-dimethyluracil

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About This Item

Empirical Formula (Hill Notation):

C₂₁H₃₁N₅O₃

CAS Number:

34661-85-3

Molecular Weight:

401.50

NACRES:

NA.77

PubChem Substance ID:

24277800

UNSPSC Code:

12352200

MDL number:

MFCD00078602

Form:

solid

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Properties

form

solid

Quality Segment

100

color

white

solubility

H₂O: 0.4 mg/mL, 0.1 M HCl: 3.8 mg/mL

SMILES string

Cl[H].COc1ccccc1N2CCN(CCCNC3=C(C)C(=O)N(C)C(=O)N3C)CC2

InChI

1S/C21H31N5O3.ClH/c1-16-19(23(2)21(28)24(3)20(16)27)22-10-7-11-25-12-14-26(15-13-25)17-8-5-6-9-18(17)29-4;/h5-6,8-9,22H,7,10-15H2,1-4H3;1H

InChI key

WAZDYFHTLYHMKO-UHFFFAOYSA-N

Gene Information

human ... ADRA1A(148), ADRA1B(147), ADRA1D(146)

Description

Application

5-Methylurapidil has been used for competitive binding in radioligand binding assays.

Biochem/physiol Actions

Selective α1A-adrenoceptor antagonist; antihypertensive.

Features and Benefits

This compound is featured on the α1-Adrenoceptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Preparation Note

5-Methylurapidil is soluble in water at 0.4 mg/ml and is also soluble in 0.1 M HCl at 3.8 mg/ml.

Storage Class

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)

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Certificates of Analysis (COA)

Lot/Batch Number

101K4608

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Articles

α1-Adrenoceptor Characteristics and Modulators

Review alpha 1 adrenoceptors as well as their agonists, antagonists, and tissue expression patterns. We suggest several modulators and alternatives for working with a-1 adrenoreceptors.

Global Trade Item Number

SKU	GTIN
EPP0625-0020-1EA	04061835083091
U101-50MG	04061832094151
U101-10MG	04061832094144

Key Documents

5-Methylurapidil

solid

Select a Size

About This Item

form

Quality Segment

color

solubility

SMILES string

InChI

InChI key

Gene Information

Application

Biochem/physiol Actions

Features and Benefits

Preparation Note

Safety Information

Storage Class

wgk

flash_point_f

flash_point_c

ppe

Documentation

Certificates of Analysis (COA)

Already Own This Product?

Protocols and Articles

Articles

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Product Citations

Global Trade Item Number