117714

应用筛选条件

关键词:'117714'

显示 1-18 共 18 条结果关于 "117714" 范围论文

[Synthesis and characterization of complex of NdL3.2H2O].

Y Yang et al.

Guang pu xue yu guang pu fen xi = Guang pu, 20(3), 322-323 (2003-09-10)

The binary solid complexes using rare earth ion Nd3+ with the ligand L (L = O-chorophenoxyacetic acid and 3-methoxybenzoic acid) has been synthesized in this work. The chemical formula of the complex was determined to be NdL3.2H2O by elemental analysis.

Antibacterial alkoxybenzamide inhibitors of the essential bacterial cell division protein FtsZ.

Lloyd G Czaplewski et al.

Bioorganic & medicinal chemistry letters, 19(2), 524-527 (2008-12-10)

3-Methoxybenzamide is a weak inhibitor of the essential bacterial cell division protein FtsZ. Exploration of the structure-activity relationships of 3-methoxybenzamide analogues led to the identification of potent anti-staphylococcal compounds.

Sodium borohydride reduction of aromatic carboxylic acids via methyl esters.

Saeed A and Ashraf Z.

Journal of Chemical Sciences (Bangalore), 118(5), 419-423 (2006)

Mass spectrometric behavior of phenolic acids standards and their analysis in the plant samples with LC/ESI/MS system.

Wojciech Ostrowski et al.

Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 967, 21-27 (2014-07-27)

Liquid chromatography coupled to mass spectrometry (MS) with electrospray ionization (ESI) is one of analytical techniques to obtain accurate results of low molecular weight aromatic compounds in biological samples of different origin. The interpretations of mass spectra of these aromatic

Toward a better understanding on the mechanism of ortholithiation. Tuning of selectivities in the metalation of meta-anisic acid by an appropriate choice of base.

Thi-Huu Nguyen et al.

Organic letters, 7(12), 2445-2448 (2005-06-04)

[reaction: see text] If employed in THF at 0 degrees C, LTMP metalates meta-anisic acid at the doubly activated position. In contrast, n-BuLi/t-BuOK deprotonates position C-4 preferentially at low temperature. Functionalization at C-6 requires protection of the C-2 site beforehand.

Hepatic microsomal thiol methyltransferase is involved in stereoselective methylation of pharmacologically active metabolite of prasugrel.

Miho Kazui et al.

Drug metabolism and disposition: the biological fate of chemicals, 42(7), 1138-1145 (2014-04-16)

Prasugrel, a thienopyridine antiplatelet drug, is converted in animals and humans to the pharmacologically active metabolite R-138727 [(2Z)-{1-[(1RS)-2-cyclopropyl-1-(2-fluorophenyl)-2-oxoethyl]-4-sulfanylpiperidin-3-ylidene}ethanoic acid], which has two chiral centers, occurring as a mixture of four isomers. The RS and RR isomers are more active than

Effects of solute characteristics and concentration on a lyotropic liquid crystal: solute-induced phase change.

H G Ibrahim et al.

Pharmaceutical research, 10(5), 737-742 (1993-05-01)

We investigated the effects of increased concentrations of the solutes, salicylic acid, benzoic acid, and o-, m-, and p-methoxy benzoic acids, on the anisotropic properties of a liquid crystal solvent. The lamellar liquid crystal was composed of 37% polyoxyethylene (20)

The versatility of the fungal cytochrome P450 monooxygenase system is instrumental in xenobiotic detoxification.

Ljerka Lah et al.

Molecular microbiology, 81(5), 1374-1389 (2011-08-04)

Cytochromes P450 (CYPs) catalyse diverse reactions and are key enzymes in fungal primary and secondary metabolism, and xenobiotic detoxification. CYP enzymatic properties and substrate specificity determine the reaction outcome. However, CYP-mediated reactions may also be influenced by their redox partners.

Stimulation of intrachromosomal homologous recombination in mammalian cells by an inhibitor of poly(ADP-ribosylation).

A S Waldman et al.

Nucleic acids research, 19(21), 5943-5947 (1991-11-11)

We determined the effect of 3-methoxybenzamide (3-MB), a competitive inhibitor of poly(ADP-ribose) polymerase (E.C. 2.4.2.30), on intrachromosomal homologous recombination in mouse Ltk- cells. We used a cell line that contained in its genome two defective Herpes thymidine kinase (tk) genes

The trans-anethole degradation pathway in an Arthrobacter sp.

Eyal Shimoni et al.

The Journal of biological chemistry, 277(14), 11866-11872 (2002-01-24)

A bacterial strain (TA13) capable of utilizing t-anethole as the sole carbon source was isolated from soil. The strain was identified as Arthrobacter aurescens based on its 16 S rRNA gene sequence. Key steps of the degradation pathway of t-anethole

Comparative functional characterization of a novel benzoate hydroxylase cytochrome P450 of Fusarium oxysporum.

Pradeepraj Durairaj et al.

Enzyme and microbial technology, 70, 58-65 (2015-02-11)

FoCYP53A19, a novel cytochrome P450 capable of performing benzoate hydroxylation, was identified and characterized from the ascomycete Fusarium oxysporum f.sp. lycopersici. Comparative functional analysis of FoCYP53A19 with the heterologous and homologous cytochrome P450 reductases (CPR) such as Saccharomyces cerevisiae (ScCPR)

Synthesis, characterization and thermal behaviour of solid-state compounds of europium (III) and gadolinium (III) 3-methoxybenzoate.

Dametto PR, et al.

Journal of Thermal Analysis and Calorimetry, 97(2), 765-768 (2009)

S-methylation of 2-mercaptopyrazine in rat liver microsomes and cytosol.

D H Lee et al.

Xenobiotica; the fate of foreign compounds in biological systems, 29(9), 909-916 (1999-11-05)

1. 2-(Allylthio)pyrazine (2-AP) has been demonstrated to protect the liver against toxicants by inhibiting CYP2E1 activity. Since 2-mercaptopyrazine (2-MP) is presumed to be a metabolite of 2-AP, the experiments were performed to determine whether rat liver microsomal and/or cytosolic preparations

3D-QSAR and molecular docking studies of benzaldehyde thiosemicarbazone, benzaldehyde, benzoic acid, and their derivatives as phenoloxidase inhibitors.

Chao-Bin Xue et al.

Bioorganic & medicinal chemistry, 15(5), 2006-2015 (2007-01-30)

Phenoloxidase (PO), also known as tyrosinase, is a key enzyme in insect development, responsible for catalyzing the hydroxylation of tyrosine into o-diphenols and the oxidation of o-diphenols into o-quinones. Inhibition of PO may provide a basis for novel environmentally friendly

Utilization of methoxylated benzoates and formation of intermediates by Desulfotomaculum thermobenzoicum in the presence or absence of sulfate.

M Tasaki et al.

Archives of microbiology, 157(3), 209-212 (1992-01-01)

Desulfotomaculum thermobenzoicum strain TSB (DSM 6193) was found to utilize some methoxylated benzoates as carbon and energy source with or without sulfate. 3- or 4-Methoxybenzoate, vanillate (4-hydroxy-3-methoxybenzoate), syringate (3,5-dimethoxy-4-hydroxybenzoate) and 3,4,5-trimethoxybenzoate were converted to corresponding hydroxybenzoates. However, neither 2-methoxybenzoate nor

Characterization of the superinduction of the c-myc proto-oncogene in fibroblasts by benzamide derivatives.

P E Devaraj et al.

Molecular and cellular biochemistry, 124(2), 175-181 (1993-07-21)

In mouse fibroblasts stimulated from quiescence into proliferation by serum the induction of expression of the c-myc proto-oncogene is strongly stimulated by 3-methoxybenzamide. Similar superinduction effects are seen with related compounds such as 3-aminobenzamide and the acid analogues, 3-anisic acid

Metabolism of the 18O-methoxy substituent of 3-methoxybenzoic acid and other unlabeled methoxybenzoic acids by anaerobic bacteria.

K A DeWeerd et al.

Applied and environmental microbiology, 54(5), 1237-1242 (1988-05-01)

O-methyl substituents of aromatic compounds can provide C1 growth substrates for facultative and strict anaerobic bacteria isolated from diverse environments. The mechanism of the bioconversion of methoxylated benzoic acids to the hydroxylated derivatives was investigated with a model substrate and

Platinum (II) complexes of benzoic- and 3-methoxybenzoic acid hydrazides. Synthesis, characterization, and cytotoxic effect.

N Dodoff et al.

Journal of inorganic biochemistry, 54(3), 221-233 (1994-05-15)

The complexes [Pt(bah)2X2], [Pt(NH3)(bah)Cl2].0.5H2O, [Pt(mbah)2X2], and [Pt(NH3)(mbah)Cl2] (bah = benzoic acid hydrazide, mbah = 3-methoxybenzoic acid hydrazide; X = Cl, Br, I) have been prepared and characterized by elemental analysis, electric conductivity, IR, 1H NMR, and electronic spectra. A cis-square

1/1