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EGFR Inhibitor
[Cyclopropanecarboxylic acid-(3-(6-(3-trifluoromethyl-phenylamino)-pyrimidin-4-
ylamino
n/d n/d
339 HDRP/MITR H9163 9734 HDAC9 P NP_001191073.1,NP_001191074.1 ,NP_001191075.1 , y y n/d
327 HDAC-4 H9411 9759 HDAC4 P NP_006028.2 y y y
328 HDAC-4 H9536 9759 HDAC4 P NP_006028.2 y y y
763 Y14
n/d n/d
339 HDRP/MITR H9163 9734 HDAC9 P NP_001191073.1,NP_001191074.1 ,NP_001191075.1 , y y n/d
327 HDAC-4 H9411 9759 HDAC4 P NP_006028.2 y y y
328 HDAC-4 H9536 9759 HDAC4 P NP_006028.2 y y y
763 Y14
n/d n/d
339 HDRP/MITR H9163 9734 HDAC9 P NP_001191073.1,NP_001191074.1 ,NP_001191075.1 , y y n/d
327 HDAC-4 H9411 9759 HDAC4 P NP_006028.2 y y y
328 HDAC-4 H9536 9759 HDAC4 P NP_006028.2 y y y
763 Y14
-1 H6287 M y y n/d
323 HDAC-2 H3159 P y y y
324 HDAC-2 H2663 M y y y
325 HDAC-3 H6537 M y y n/d
326 HDAC-3 H3034 P y y y
327 HDAC-4 H9411 P y y y
328 HDAC-4 H9536 P y
.2 M y y y
325 HDAC-3 H6537 15183, 8841 Hdac3,HDAC3 NP_034541.2,NP_003874.2 M y y n/d
326 HDAC-3 H3034 15183, 8841, 84578 Hdac3,HDAC3 NP_034541.2,NP_003874.2,NP_445900.1 P y y y
327 HDAC-4 H9411 208727
.2 M y y y
325 HDAC-3 H6537 15183, 8841 Hdac3,HDAC3 NP_034541.2,NP_003874.2 M y y n/d
326 HDAC-3 H3034 15183, 8841, 84578 Hdac3,HDAC3 NP_034541.2,NP_003874.2,NP_445900.1 P y y y
327 HDAC-4 H9411 208727
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327
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