371725
GPR43 Agonist
>98% (HPLC), solid
别名:
GPR43（FFA2）激动剂, （S）-2-（4-氯苯基）-3，3-二甲基-N-（5-苯基噻唑-2-基）丁酰胺
产品名称
GPR43（FFA2）激动剂, The GPR43 (FFA2) Agonist controls the biological activity of GPR43. This small molecule/inhibitor is primarily used for Biochemicals applications.
质量水平
方案
>98% (HPLC)
表单
solid
制造商/商品名称
Calbiochem®
储存条件
OK to freeze
颜色
white
溶解性
DMSO: 50 mg/mL
运输
ambient
储存温度
2-8°C
一般描述
一种苯乙酰胺化合物，可作为FFA2的变构激动剂（GPR43），在hFFA2毛喉素诱导的cAMP分析中显示出相对于乙酸盐的左移乙酸盐剂量反应（IC50 = 0.7 µM）和111%的功效。
制备说明
复溶后，等分并冷冻保存（-20°C）。储备溶液在-20°C下可稳定保存至多3个月。
其他说明
Wang, Y., et al. 2009.Bioorg.Med. Chem. Lett.20, 493.
法律信息
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
免责声明
毒性：标准处理（A）
储存分类代码
11 - Combustible Solids
WGK
WGK 3
闪点(°F)
Not applicable
闪点(°C)
Not applicable
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