371725
GPR43 Agonist
>98% (HPLC), solid
别名:
GPR43（FFA2）激动剂, （S）-2-（4-氯苯基）-3，3-二甲基-N-（5-苯基噻唑-2-基）丁酰胺
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关于此项目
经验公式（希尔记法）:
C21H21ClN2OS
化学文摘社编号:
分子量:
384.92
MDL number:
UNSPSC Code:
51111800
NACRES:
NA.77
产品名称
GPR43（FFA2）激动剂, The GPR43 (FFA2) Agonist controls the biological activity of GPR43. This small molecule/inhibitor is primarily used for Biochemicals applications.
assay
>98% (HPLC)
form
solid
manufacturer/tradename
Calbiochem®
storage condition
OK to freeze
color
white
solubility
DMSO: 50 mg/mL
shipped in
ambient
Quality Level
相关类别
General description
一种苯乙酰胺化合物，可作为FFA2的变构激动剂（GPR43），在hFFA2毛喉素诱导的cAMP分析中显示出相对于乙酸盐的左移乙酸盐剂量反应（IC50 = 0.7 µM）和111%的功效。
Preparation Note
复溶后，等分并冷冻保存（-20°C）。储备溶液在-20°C下可稳定保存至多3个月。
Other Notes
Wang, Y., et al. 2009.Bioorg.Med. Chem. Lett.20, 493.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Disclaimer
毒性：标准处理（A）
存储类别
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
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