5.05878
PD 168077 Maleate
别名:
PD 168077 Maleate, D4 Dopamine Receptor Agonist, PD 168077 Maleate, PD168077, PD-168077
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关于此项目
经验公式（希尔记法）:
C20H22N4O · xC4H4O4
化学文摘社编号:
分子量:
334.41 (free base basis)
MDL number:
UNSPSC Code:
12352200
NACRES:
NA.77
SMILES string
N2(CCN(CC2)c3c(cccc3)C#N)CNC(=O)c1cc(ccc1)C.OC(=O)\C=C/C(=O)O
InChI
1S/C20H22N4O.C4H4O4/c1-16-5-4-7-17(13-16)20(25)22-15-23-9-11-24(12-10-23)19-8-3-2-6-18(19)14-21;5-3(6)1-2-4(7)8/h2-8,13H,9-12,15H2,1H3,(H,22,25);1-2H,(H,5,6)(H,7,8)/b;2-1-
InChI key
NAEUGRPISCANHO-BTJKTKAUSA-N
assay
≥98% (HPLC)
form
solid
manufacturer/tradename
Calbiochem®
storage condition
OK to freeze, protect from light
color
white
solubility
DMSO: 100 mM
storage temp.
−20°C
Quality Level
General description
A selective D4 dopamine receptor agonist (Ki = 8.7 nM, EC50 = 8.3 nM). Suitable for central and peripheral delivery. Used in studies of penile erection, learning and memory. Exibits some binding affinity towards human D2 and D3 Receptors (Ki = 2.8 µM).
Biochem/physiol Actions
Primary Target
D₄
D₄
Reversible: yes
Preparation Note
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Other Notes
Melis, M. R. et al. 2005. Neurosci. Lett.379, 59.
Bernaerts, P. et al. 2003. Behav. Brain Res.142, 41.
Bernaerts, P. et al. 2003. Behav. Brain Res.142, 41.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Disclaimer
Toxicity: Standard Handling (A)
存储类别
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
法规信息
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