BM0014
BMS-207940
≥98% (HPLC)
别名:
Edonentan, N-[[2′-[[(4,5-Dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1′-biphenyl]-2-yl]methyl]-N,3,3-trimethylbutanamide
方案
≥98% (HPLC)
表单
powder
颜色
white to beige
溶解性
DMSO: 20 mg/mL, clear
储存温度
room temp
SMILES字符串
O=S(NC1=NOC(C)=C1C)(C2=C(C3=CC=C(C4=NC=CO4)C=C3CN(C)C(CC(C)(C)C)=O)C=CC=C2)=O
InChI
1S/C28H32N4O5S/c1-18-19(2)37-30-26(18)31-38(34,35)24-10-8-7-9-23(24)22-12-11-20(27-29-13-14-36-27)15-21(22)17-32(6)25(33)16-28(3,4)5/h7-15H,16-17H2,1-6H3,(H,30,31)
InChI key
ORJRYNKVKJAJPY-UHFFFAOYSA-N
生化/生理作用
BMS-207940 is a very potent and selective ETA endothelin receptor antagonist.
BMS-207940 is a very potent and selective ETA endothelin receptor antagonist. BMS-207940 has a Ki of 10 pM for ETA, 80000-fold selective for ETA vs ETB.
特点和优势
BMS-207940 is available through a partnership with Bristol-Myers Squibb (BMS). To learn more and view other BMS compounds, visit sigma.com/BMS.
法律信息
Sold for research purposes only under agreement from BMS.
储存分类代码
13 - Non Combustible Solids
WGK
WGK 3
闪点(°F)
Not applicable
闪点(°C)
Not applicable
法规信息
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