Fluorescent Adenosine receptor Antagonist (A-633-AN) synthetic

The SML0156 ligand was shown to antagonize the activity of the adenosine receptor agonist adenosine-5′-N-ethyluronamide (NECA), in three separate recombinant CHO cell lines expressing the human A1, A2A or A3 receptor and a cyclic AMP-responsive secreted placental alkaline phosphatase (SPAP) reporter gene.

This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Dissolve 0.2 mg in 20.5 ul of DMSO to give a 10mM stock solution. Once reconstituted into DMSO the product, must be stored, preferably in smaller aliquots, at -20°C.