V5390
VU0029251
≥98% (HPLC), powder
别名:
6,7-Dihydro-2-(methylthio)-5H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-4-amine
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关于此项目
经验公式（希尔记法）:
C10H11N3S2
分子量:
237.34
MDL编号:
UNSPSC代码:
12352200
PubChem化学物质编号:
NACRES:
NA.77
方案
≥98% (HPLC)
表单
powder
颜色
white to tan
溶解性
DMSO: ≥11 mg/mL
储存温度
2-8°C
SMILES字符串
CSc1nc(N)c2c3CCCc3sc2n1
InChI
1S/C10H11N3S2/c1-14-10-12-8(11)7-5-3-2-4-6(5)15-9(7)13-10/h2-4H2,1H3,(H2,11,12,13)
InChI key
WDDBZCKBRCTSOZ-UHFFFAOYSA-N
生化/生理作用
VU0029251 is the first example of a partial mGluR5 partial antagonist that is not based on the MPEP scaffold.
VU0029251 is the first example of a partial mGluR5 partial antagonist that is not based on the MPEP scaffold. The compound displays a maximum inhibition of 50% activity, and cannot completely displace [3H] MPEP, suggesting that competition for MPEP is also allosteric, involving a unique site.
特点和优势
This compound is featured on the Glutamate Receptors (G Protein Family) page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
储存分类代码
13 - Non Combustible Solids
WGK
WGK 3
闪点(°F)
Not applicable
闪点(°C)
Not applicable
法规信息
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